Synthesis of a novel family of diterpenes and their evaluation as anti-inflammatory agents.

نویسندگان

  • Thanh Lam
  • Taotao Ling
  • Chinmay Chowdhury
  • Ta-Hsiang Chao
  • F R Bahjat
  • G K Lloyd
  • Lyle L Moldawer
  • Michael A Palladino
  • Emmanuel A Theodorakis
چکیده

The synthesis and biological evaluation of a new family of diterpenes, represented by structures 2 and 3, is presented. These compounds constitute isomeric analogues of acanthoic acid (1) and were examined as potent anti-inflammatory agents. Among them, methyl ester 12 exhibited a low non-specific cytotoxicity, inhibited TNF-alpha synthesis and displayed good specificity in suppressing cytokine expression.

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عنوان ژورنال:
  • Bioorganic & medicinal chemistry letters

دوره 13 19  شماره 

صفحات  -

تاریخ انتشار 2003